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perlapine

perlapine Structural

What is perlapine?

The Uses of perlapine

Perlapine is an atypical neuroleptic that blocks dopamine and serotonin (5-HT) receptors (Kis = 60, 30, and 30 nM for D2, D4, and 5-HT2A, respectively). Perlapine is also an agonist for hM3Dq, a designer receptor exclusively activated by designer drugs (DREADD) derived from the human muscarinic acetylcholine M3 receptor that activates neuronal firing. Perlapine displays >10,000-fold selectivity for hM3Dq over hM3.

The Uses of perlapine

Perlapine exhibits antipsychotic activity and blocks dopamine and serotonin receptors. Perlapine is also a novel agonist of hM3Dq, a designer receptor exclusively activated by designer drugs (DREADD).

Definition

ChEBI: Perlapine is an organic molecular entity.

storage

Room temperature

Properties of perlapine

Melting point: 136-138°
Boiling point: 423.4°C (rough estimate)
Density  1.0521 (rough estimate)
refractive index  1.6080 (estimate)
storage temp.  Store at -20°C
solubility  DMF: 10 mg/ml; DMSO: 10 mg/ml; DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml; Ethanol: 5 mg/ml
form  A crystalline solid
pka 8.00±0.20(Predicted)
color  White

Safety information for perlapine

Computed Descriptors for perlapine

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