MRS 1706
Synonym(s):8-[4-[((4-Acetylphenyl)carbamoylmethyl)oxy]phenyl]-1,3-di(n-propyl)xanthine;MRS 1706;MRS1706;N-(4-Acetylphenyl)-2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,9-tetrahydro-1H-purin-8-yl)phenoxy)acetamide;N-(4-Acetylphenyl)-2-[4-(2,3,6,9-tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl)phenoxy]acetamide
- CAS NO.:264622-53-9
- Empirical Formula: C27H29N5O5
- Molecular Weight: 503.55
- MDL number: MFCD28160689
- SAFETY DATA SHEET (SDS)
- Update Date: 2024-11-09 21:40:10
What is MRS 1706?
Description
MRS1706 is a selective adenosine A2B receptor inverse agonist with Ki values of 1.39, 157, 112, and 230 nM for human A2B, A1, A2A, and A3 receptors, respectively.
The Uses of MRS 1706
MRS 1706 is a selective and potent Adenosine A2B-R inverse agonist Ki (binding affinity) values of 1.39, 157, 112, and 230 nM for human A2B, A1, A2A, and A3 receptors, respectively.
What are the applications of Application
MRS 1706 is a selective and potent Adenosine A2B-R inverse agonist
Biological Activity
Potent and selective adenosine A 2B receptor inverse agonist (K i values are 1.39, 157, 112 and 230 nM for human A 2B , A 1 , A 2A and A 3 receptors respectively).
Properties of MRS 1706
Density | 1.293±0.06 g/cm3(Predicted) |
storage temp. | Sealed in dry,2-8°C |
solubility | DMSO : 6.4 mg/mL (12.71 mM; Need ultrasonic and warming)H2O : < 0.1 mg/mL (insoluble) |
form | Powder |
pka | 8.25±0.70(Predicted) |
color | Off-white to yellow |
Safety information for MRS 1706
Computed Descriptors for MRS 1706
New Products
ALUMINIUM IODIDE 100 GM BUFFER CAPSULE PH 7.0 - 10 CAP BUFFER SOLUTION PH 9.5 (BORATE) EZEE BLUE GEL STAINER BORAX CARMINE (GRENACHERS ALCOHOLIC) POTASSIUM IODATE - IODIDE SOLN 0.1 N Dabigatran Acyl-O3-D-Glucuronide Trifluoroacetic Acid Salt Isofolic Acid Dabigatran 2-O-acylglucuronide metabolite Dabigatran Acyl-?-D- glucuronide Trifluroacetic Acid Erythromycin EP Impurity A Desloratidine Related Compound ARelated products of tetrahydrofuran
1,3-DIETHYL-8-PHENYLXANTHINE
MRS 1706
8-PHENYLTHEOPHYLLINE
1,3-DIPROPYL-8-PHENYLXANTHINE
2-(4-ETHOXY-PHENYL)-1H-IMIDAZOLE
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