MRS 1220
Synonym(s):9-Chloro-2-(2-furanyl)-5-((phenylacetyl)amino)-[1,2,4]triazolo[1,5-c]quinazoline
- CAS NO.：183721-15-5
- Empirical Formula: C21H14ClN5O2
- Molecular Weight: 403.82
- MDL number: MFCD01321046
- SAFETY DATA SHEET (SDS)
- Update Date: 2024-11-19 23:02:33
What is MRS 1220?
The Uses of MRS 1220
MRS 1220 is a highly potent and selective human Adenosine A3-R antagonist.
What are the applications of Application
MRS 1220 is a highly potent and selective human Adenosine A3-R antagonist
Definition
ChEBI: N-[9-chloro-2-(2-furanyl)-[1,2,4]triazolo[1,5-c]quinazolin-5-yl]-2-phenylacetamide is a member of quinazolines.
Biological Activity
A potent and highly selective antagonist at the human A 3 adenosine receptor (K i values are 0.65, 305, and 52 nM at hA 3 , rA 1 and rA 2A respectively. Displays an IC 50 value > 1 μ M for inhibition of binding to rat A 3 receptors).
storage
Store at RT
Properties of MRS 1220
| Density | 1.49±0.1 g/cm3(Predicted) |
| storage temp. | Store at RT |
| solubility | DMSO: 2 mg/mL |
| form | solid |
| pka | 8.17±0.46(Predicted) |
| color | white |
Safety information for MRS 1220
Computed Descriptors for MRS 1220
New Products
(S)-3-Aminobutanenitrile hydrochloride 4-Methylphenylacetic acid N-Boc-D-alaninol N-BOC-D/L-ALANINOL Tert-butyl bis(2-chloroethyl)carbamate 3-Morpholino-1-(4-nitrophenyl)-5,6-dihydropyridin- 2(1H)-one Furan-2,5-Dicarboxylic Acid Tropic acid 1-Bromo-3,5-Di-Tert-Butylbenzene S-2-CHLORO PROPIONIC ACID ETHYL ISOCYANOACETATE 2-Bromo-1,3-Bis(Dimethylamino)Trimethinium Hexafluorophosphate 4-IODO BENZOIC ACID 3-NITRO-2-METHYL ANILINE 1-(2,4-DICHLOROPHENYL) ETHANAMINE (2-Hydroxyphenyl)acetonitrile 4-Bromopyrazole 2-(Cyanocyclohexyl)acetic acid 4-methoxy-3,5-dinitropyridine 1-(4-(aminomethyl)benzyl)urea hydrochloride 2-aminopropyl benzoate hydrochloride diethyl 2-(2-((tertbutoxycarbonyl)amino) ethyl)malonate tert-butyl 4- (ureidomethyl)benzylcarbamate Ethyl-2-chloro((4-methoxyphenyl)hydrazono)acetateRelated products of tetrahydrofuran
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